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ONC-ORG

Cancer Drug Encyclopedia

Approved oncology medications — what they treat, how they work and key safety information.

XatmepMethotrexate Sodium
Cytotoxic Antimetabolite Chemotherapeutic AgentLyophilized Powder / Solution for Intravenous Infusion

Colorectal, Pancreatic, Breast, Non-Small Cell Lung Cancer, Myelodysplastic Syndromes (MDS), and Acute/Chronic Leukemias.

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XelodaCapecitabine
Cytotoxic Antimetabolite Chemotherapeutic AgentOral Film-Coated Tablet

Colorectal, Pancreatic, Breast, Non-Small Cell Lung Cancer, Myelodysplastic Syndromes (MDS), and Acute/Chronic Leukemias.

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XgevaDenosumab
Targeted Monoclonal AntibodyIntravenous Solution / Subcutaneous Injection

Targeted treatment of solid tumors and hematologic malignancies.

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XofigoRadium 223 Dichloride
Targeted Radiopharmaceutical / Radioligand TherapySingle-dose Intravenous Radioactive Solution

PSMA-positive Metastatic Castration-Resistant Prostate Cancer, Gastroenteropancreatic Neuroendocrine Tumors (GEP-NETs), and Pheochromocytoma.

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XospataGilteritinib Fumarate
Targeted Small Molecule Kinase InhibitorOral Film-Coated Tablet / Capsule

Advanced solid tumors and hematologic malignancies with matching genomic alterations.

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XpovioSelinexor
Targeted Oncology AgentOral Tablet / Capsule

Approved for use in oncology care according to FDA-approved indications.

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Xtandienzalutamide
Androgen Receptor Inhibitor (Antiandrogen)Oral Tablet / Capsule

Treatment of patients with castration-resistant prostate cancer (CRPC) and metastatic castration-sensitive prostate cancer (mCSPC).

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YervoyIpilimumab
Immune Checkpoint Inhibitor (PD-1 / PD-L1 / CTLA-4)Intravenous Solution / Subcutaneous Injection

Melanoma, Non-Small Cell Lung Cancer, Renal Cell Carcinoma, Urothelial Cancer, Head and Neck Cancer, MSI-H/dMMR solid tumors, and Cervical Cancer.

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YescartaAxicabtagene Ciloleucel
Autologous CAR T-Cell ImmunotherapySingle-dose Intravenous Suspension for Infusion

Relapsed or refractory B-cell Acute Lymphoblastic Leukemia, Large B-cell Lymphoma, Mantle Cell Lymphoma, or Multiple Myeloma.

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YondelisTrabectedin
Targeted Oncology AgentOral Tablet / Capsule

Approved for use in oncology care according to FDA-approved indications.

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YonsaAbiraterone Acetate
CYP17 Inhibitor / Androgen Biosynthesis InhibitorOral Tablet (taken on an empty stomach)

Metastatic Castration-Resistant Prostate Cancer (mCRPC) and High-Risk Castration-Sensitive Prostate Cancer in combination with prednisone.

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ZaltrapZiv-Aflibercept
Targeted Oncology AgentOral Tablet / Capsule

Approved for use in oncology care according to FDA-approved indications.

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