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ONC-ORG

Cancer Drug Encyclopedia

Approved oncology medications — what they treat, how they work and key safety information.

LutatheraLutetium Lu 177-Dotatate
Targeted Radiopharmaceutical / Radioligand TherapySingle-dose Intravenous Radioactive Solution

PSMA-positive Metastatic Castration-Resistant Prostate Cancer, Gastroenteropancreatic Neuroendocrine Tumors (GEP-NETs), and Pheochromocytoma.

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LutetiumLu 177-Dotatate
Targeted Radiopharmaceutical / Radioligand TherapySingle-dose Intravenous Radioactive Solution

PSMA-positive Metastatic Castration-Resistant Prostate Cancer, Gastroenteropancreatic Neuroendocrine Tumors (GEP-NETs), and Pheochromocytoma.

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Lutetium Lu 177 Vipivotide TetraxetanLutetium Lu 177 Vipivotide Tetraxetan
Targeted Radiopharmaceutical / Radioligand TherapySingle-dose Intravenous Radioactive Solution

PSMA-positive Metastatic Castration-Resistant Prostate Cancer, Gastroenteropancreatic Neuroendocrine Tumors (GEP-NETs), and Pheochromocytoma.

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LymphirDenileukin Diftitox-cxdl
Targeted Oncology AgentOral Tablet / Capsule

Approved for use in oncology care according to FDA-approved indications.

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Lynparzaolaparib
Poly (ADP-ribose) Polymerase (PARP) InhibitorOral Tablet / Capsule

Maintenance treatment of adult patients with deleterious or suspected deleterious germline or somatic BRCA-mutated advanced ovarian, breast, pancreatic, and prostate cancer.

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LytgobiFutibatinib
Targeted Small Molecule Kinase InhibitorOral Film-Coated Tablet / Capsule

Advanced solid tumors and hematologic malignancies with matching genomic alterations.

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MOPPMechlorethamine, Vincristine, Procarbazine, Prednisone
Historical Alkylating RegimenMulti-agent Intravenous Chemotherapy Protocol

Historic first-line treatment for Hodgkin Lymphoma (now primarily used in specific relapsed settings).

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MVACMethotrexate, Vinblastine, Doxorubicin, Cisplatin
Urothelial Cancer Chemotherapy RegimenMulti-agent Intravenous Chemotherapy Protocol

Locally advanced or metastatic Bladder / Urothelial Carcinoma.

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MargenzaMargetuximab-cmkb
HER2-Directed Monoclonal AntibodyIntravenous Solution / Subcutaneous Injection

HER2-overexpressing Breast Cancer, metastatic Gastric Cancer, and gastroesophageal junction adenocarcinoma.

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Margetuximab-cmkbMargetuximab-cmkb
HER2-Directed Monoclonal AntibodyIntravenous Solution / Subcutaneous Injection

HER2-overexpressing Breast Cancer, metastatic Gastric Cancer, and gastroesophageal junction adenocarcinoma.

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MatulaneProcarbazine Hydrochloride
DNA Alkylating Chemotherapeutic AgentOral Capsule

Brain Tumors (Glioblastoma, Astrocytoma), Multiple Myeloma, Lymphomas, Leukemias, Sarcomas, and conditioning regimens.

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Mechlorethamine HydrochlorideMechlorethamine Hydrochloride
Targeted Oncology AgentOral Tablet / Capsule

Approved for use in oncology care according to FDA-approved indications.

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