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Cancer Drug Encyclopedia

Approved oncology medications — what they treat, how they work and key safety information.

Acalabrutinib Maleate MonohydrateAcalabrutinib Maleate Monohydrate
Bruton's Tyrosine Kinase (BTK) InhibitorOral Film-Coated Tablet / Capsule

Chronic Lymphocytic Leukemia (CLL), Small Lymphocytic Lymphoma (SLL), Mantle Cell Lymphoma, Waldenström's Macroglobulinemia.

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ActemraTocilizumab
Targeted Monoclonal AntibodyIntravenous Solution / Subcutaneous Injection

Targeted treatment of solid tumors and hematologic malignancies.

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AdagrasibAdagrasib
KRAS G12C Specific InhibitorOral Film-Coated Tablet / Capsule

KRAS G12C-mutated Non-Small Cell Lung Cancer and advanced Colorectal Cancer.

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AdcetrisBrentuximab Vedotin
Targeted Antibody-Drug Conjugate (ADC)Lyophilized Powder for Intravenous Infusion

Hodgkin Lymphoma, CD30-expressing T-cell lymphomas, Urothelial Carcinoma, Cervical Cancer, or Diffuse Large B-cell Lymphoma.

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Ado-Trastuzumab EmtansineAdo-Trastuzumab Emtansine
Targeted Antibody-Drug Conjugate (ADC)Lyophilized Powder for Intravenous Infusion

HER2-positive or HER2-low metastatic Breast Cancer, HER2-mutant Non-Small Cell Lung Cancer, and Gastric Adenocarcinoma.

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AdriamycinDoxorubicin Hydrochloride
Topoisomerase Inhibitor Chemotherapy AgentIntravenous Solution for Infusion

Breast Cancer, Small Cell Lung Cancer, Colorectal Cancer, Ovarian Cancer, and Acute Leukemias.

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AdstiladrinNadofaragene Firadenovec-vncg
Targeted Oncology AgentOral Tablet / Capsule

Approved for use in oncology care according to FDA-approved indications.

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Afamitresgene AutoleucelAfamitresgene Autoleucel
Autologous CAR T-Cell ImmunotherapySingle-dose Intravenous Suspension for Infusion

Relapsed or refractory B-cell Acute Lymphoblastic Leukemia, Large B-cell Lymphoma, Mantle Cell Lymphoma, or Multiple Myeloma.

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Afatinib DimaleateAfatinib Dimaleate
EGFR Tyrosine Kinase InhibitorOral Film-Coated Tablet / Capsule

EGFR-mutated Non-Small Cell Lung Cancer (NSCLC).

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AfinitorEverolimus
Targeted Oncology AgentOral Tablet / Capsule

Approved for use in oncology care according to FDA-approved indications.

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AkeegaNiraparib Tosylate Monohydrate and Abiraterone Acetate
Poly (ADP-ribose) Polymerase (PARP) InhibitorOral Tablet / Capsule

Deleterious BRCA-mutated or HRD-positive Ovarian, Breast, Pancreatic, and Prostate Cancers.

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AkynzeoNetupitant and Palonosetron Hydrochloride
Antiemetic Supportive Agent (5-HT3 / NK1 Receptor Antagonist)Oral Tablet / Intravenous Solution

Prevention and management of chemotherapy-induced and radiation-induced nausea and vomiting (CINV).

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