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ONC-ORG

Cancer Drug Encyclopedia

Approved oncology medications — what they treat, how they work and key safety information.

TolakFluorouracil Topical
Cytotoxic Antimetabolite Chemotherapeutic AgentTopical Cream / Solution (0.5% - 5%)

Colorectal, Pancreatic, Breast, Non-Small Cell Lung Cancer, Myelodysplastic Syndromes (MDS), and Acute/Chronic Leukemias.

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Topotecan HydrochlorideTopotecan Hydrochloride
Topoisomerase Inhibitor Chemotherapy AgentIntravenous Solution for Infusion

Breast Cancer, Small Cell Lung Cancer, Colorectal Cancer, Ovarian Cancer, and Acute Leukemias.

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ToremifeneToremifene
Selective Estrogen Receptor Modulator / Degrader (SERM/SERD)Oral Tablet

HR-positive Breast Cancer in adjuvant, metastatic, and chemoprevention settings.

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Toripalimab-tpziToripalimab-tpzi
Immune Checkpoint Inhibitor (PD-1 / PD-L1 / CTLA-4)Intravenous Solution / Subcutaneous Injection

Melanoma, Non-Small Cell Lung Cancer, Renal Cell Carcinoma, Urothelial Cancer, Head and Neck Cancer, MSI-H/dMMR solid tumors, and Cervical Cancer.

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ToriselTemsirolimus
Targeted Oncology AgentOral Tablet / Capsule

Approved for use in oncology care according to FDA-approved indications.

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TotectDexrazoxane Hydrochloride
Oncology Supportive / Cytoprotective AgentIntravenous Solution

Prevention and management of chemotherapy-related organ toxicities and complications.

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TovorafenibTovorafenib
BRAF / MEK Kinase InhibitorOral Film-Coated Tablet / Capsule

BRAF V600E/K mutation-positive Melanoma, Non-Small Cell Lung Cancer, Anaplastic Thyroid Cancer, and Colorectal Cancer.

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TrabectedinTrabectedin
Targeted Oncology AgentOral Tablet / Capsule

Approved for use in oncology care according to FDA-approved indications.

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Trametinib Dimethyl SulfoxideTrametinib Dimethyl Sulfoxide
BRAF / MEK Kinase InhibitorOral Film-Coated Tablet / Capsule

BRAF V600E/K mutation-positive Melanoma, Non-Small Cell Lung Cancer, Anaplastic Thyroid Cancer, and Colorectal Cancer.

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TrastuzumabTrastuzumab
HER2-Directed Monoclonal AntibodyIntravenous Solution / Subcutaneous Injection

HER2-overexpressing Breast Cancer, metastatic Gastric Cancer, and gastroesophageal junction adenocarcinoma.

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Trastuzumab and Hyaluronidase-oyskTrastuzumab and Hyaluronidase-oysk
HER2-Directed Monoclonal AntibodyIntravenous Solution / Subcutaneous Injection

HER2-overexpressing Breast Cancer, metastatic Gastric Cancer, and gastroesophageal junction adenocarcinoma.

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TreandaBendamustine Hydrochloride
DNA Alkylating Chemotherapeutic AgentIntravenous Infusion

Brain Tumors (Glioblastoma, Astrocytoma), Multiple Myeloma, Lymphomas, Leukemias, Sarcomas, and conditioning regimens.

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